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Covers the methodology for the detection and assessment of constitutively active proteins.
List of contents
Section I-- Identification and Measurement of Constitutive Activity
- Constitutive activity at the cannabinoid CB1 receptor and behavioral responses
Katherine E. Hanlon and Todd W. Vanderah
- Detecting constitutive activity and protean agonism at the cannabinoid-2 receptor.
Massimiliano Beltramo, Rossella Brusa, Isabella Mancini, Paola Scandroglio, Massimiliano. Beltramo
- Modulation of constitutive activity of the ghrelin receptor by use of pharmacological tools as well as mutagenesis
Birgitte Holst and Jacek Mokrosinski
- Assessment of constitutive activity and internalization of GPR54 (Kiss1-r).
Macarena Pampillo and Andy Videsh Babwah
- Assessment of Constitutive Activity in EP Prostanoid Receptors
Hiromichi Fujino, Toshihiko Murayama, and John W. Regan
- ?1D-Adrenergic receptors: constitutive activity and reduced expression at the plasma membrane
J Adolfo Garcia-Sáinz, M. Teresa Romero-Ávila and Luz del Carmen Medina
- Constitutive activity of the histamine H1 receptor
Saskia Nijmeijer, Rob Leurs and Henry F Vischer
- Constitutive activity of somatostatin receptor subtypes
Anat Ben-Shlomo, Kolja Wawrowsky and Shlomo Melmed
- Assessment of homologous internalization of constitutively active N111G mutant of AT1 receptor
Mohiuddin Ahmed Bhuiyan and Takafumi Nagatomo
- Methods to detect cell surface expression and constitutive activity of GPR6
Balakrishna M. Prasad, Bettye Hollins and Nevin A. Lambert
- ?3-adrenoceptor agonists and (antagonists as) inverse agonists: history, perspective, constitutive activity and stereospecific binding.
Maria Grazia Perrone and Antonio Scilimati
- Constitutive Activity of the Lutropin Receptor and its Allosteric Modulation by Receptor Heterodimerization
Deborah L. Segaloff
- Assessing Constitutive Activity of Extracellular Calcium-Sensing Receptors in Vitro and in Bone
Wenhan Chang, Melita Dvorak, and Dolores Shoback
- Constitutive Activity of Neural Melanocortin Receptors.
Ya-Xiong Tao, Hui Huang, Zhi-Qiang Wang, Fan Yang, Jessica N. Williams, and Gregory V. Nikiforovich
- Measurement of Constitutive Activity of BMP Type I receptors
Peter ten Dijke
- Probing the CA among dopamine D1 and D5 receptors and their mutants
Bianca Plouffe, Jean-Philippe D'Aoust, Vincent Laquerre, Binhui Liang and Mario Tiberi
- Identification of Gain-of-Function Variants of the Human Prolactin Receptor
Vincent Goffin, Roman L. Bogorad, and Philippe Touraine
- Investigations of Activated ACVR1/ALK2, a Bone Morphogenetic Protein (BMP) Type I Receptor that Causes Fibrodysplasia Ossificans Progressiva
Frederick. Kaplan, Petra Seemann, Julia Haupt, Meiqi Xu, Vitali Lounev, Mary Mullins, Eileen M. Shore
- Identification and evaluation of constitutively active thyroid stimulating hormone receptor mutations
Joaquin Lado-Abeal, Leah R. Quisenberry, and Isabel Castro-Piedras
- Assessment of constitutive activity of a G protein-coupled receptor, Cpr2, in Cryptococcus neoformans by heterologous and homologous methods
Chaoyang Xue, Yina Wang, and Yen-Ping Hsueh
- In vitro and in vivo assessment of mu opioid receptor constitutive activity.
Edward J. Bilsky, Denise Giuvelis, Melissa D. Osborn, Christina M. Dersch, Heng Xu and Richard B. Rothman
- Constitutively active µ-opioid methods
Mark. Connor and John Traynor
- Protein Kinase Ck2 is a Constitutively-Active Enzyme That Promotes Cell Survival: Strategies To Identify Ck2 Substrates and Manipulate Its Activity In Mammalian Cells
Jacob P. Turowec, James S. Duncan, Ashley C. French, Laszlo Gyenis, Ni
